Sciact
  • EN
  • RU

(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling Full article

Journal ACS Infectious Diseases
ISSN: 2373-8227
Output data Year: 2024, Volume: 10, Number: 6, Pages: 2127-2150 Pages count : 24 DOI: 10.1021/acsinfecdis.4c00136
Authors Golovina Anastasia 3 , Proia Eleonora 1 , Fiorentino Francesco 2 , Yunin Maxim 3 , Kasatkina Maria 3 , Zigangirova Nailya 4 , Soloveva Anna 4 , Sysolyatina Elena 4 , Ermolaeva Svetlana 4 , Novikov Roman 5 , Silonov Sergei 3 , Pushkin Sergei 3 , Mladenović Milan 6 , Isakova Julia 3 , Belik Albina 3 , Nawrozkij Maxim 3 , Rotili Dante 2 , Ragno Rino 2 , Ivanov Roman 1
Affiliations
1 Rome Center for Molecular Design, Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome 00185, Italy
2 Department of Drug Chemistry and Technologies, Sapienza University of Rome, Rome 00185, Italy;
3 Sirius University of Science and Technology, Sirius, Krasnodar Region 354340, Russia
4 National Research Centre of Epidemiology and Microbiology named after N. F. Gamaleya, Russian Health Ministry, 123098 Moscow, Russia
5 Engelhardt Institute of Molecular Biology of the Russian Academy of Sciences, Moscow 119991, Russia
6 Kragujevac Center for Computational Biochemistry, Department of Chemistry, Faculty of Science, University of Kragujevac, Kragujevac 34000, Serbia;
Cite: Golovina A. , Proia E. , Fiorentino F. , Yunin M. , Kasatkina M. , Zigangirova N. , Soloveva A. , Sysolyatina E. , Ermolaeva S. , Novikov R. , Silonov S. , Pushkin S. , Mladenović M. , Isakova J. , Belik A. , Nawrozkij M. , Rotili D. , Ragno R. , Ivanov R.
(Heteroarylmethyl)benzoic Acids as a New Class of Bacterial Cystathionine γ-Lyase Inhibitors: Synthesis, Biological Evaluation, and Molecular Modeling
ACS Infectious Diseases. 2024. V.10. N6. P.2127-2150. DOI: 10.1021/acsinfecdis.4c00136 WOS Scopus РИНЦ OpenAlex
Identifiers:
Web of science: WOS:001228938600001
Scopus: 2-s2.0-85194084452
Elibrary: 67612522
OpenAlex: W4398156415
Citing:
DB Citing
OpenAlex 1
Altmetrics: